H4 Receptor antagonist 1 ( —— )

Catalog No. M20493 CAS No. 848217-00-5

H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist with an IC50?of 19 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
2MG	40	In Stock
5MG	65	In Stock
10MG	102	In Stock
25MG	197	In Stock
50MG	356	In Stock
100MG	533	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

Product Name

H4 Receptor antagonist 1
Note

Research use only not for human use.
Brief Description

H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist with an IC50?of 19 nM.
Description

H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist with an IC50?of 19 nM.
Synonyms

——
Pathway

GPCR/G Protein
Target

Histamine Receptor
Recptor

H4 receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

848217-00-5
Formula Weight

316.78
Molecular Formula

C16H17ClN4O
Purity

>98% (HPLC)
Solubility

DMSO:10 mg/mL (31.57 mM)
SMILES

CN1CCN(CC1)c1nc(C)nc2c3cc(Cl)ccc3oc12
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Cramp S Dyke H J Higgs C et al. Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists[J]. Bioorganic & Medicinal Chemistry Letters 2010 20(8):2516-2519.

Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog

Product			Quantity Required*
Name *			E-mail Address *
Organization *			Phone Number
Remarks