H4 Receptor antagonist 1

CAS No. 848217-00-5

H4 Receptor antagonist 1 ( —— )

Catalog No. M20493 CAS No. 848217-00-5

H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist with an IC50?of 19 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 40 In Stock
5MG 65 In Stock
10MG 102 In Stock
25MG 197 In Stock
50MG 356 In Stock
100MG 533 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    H4 Receptor antagonist 1
  • Note
    Research use only not for human use.
  • Brief Description
    H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist with an IC50?of 19 nM.
  • Description
    H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist with an IC50?of 19 nM.
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    H4 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    848217-00-5
  • Formula Weight
    316.78
  • Molecular Formula
    C16H17ClN4O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mg/mL (31.57 mM)
  • SMILES
    CN1CCN(CC1)c1nc(C)nc2c3cc(Cl)ccc3oc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Cramp S Dyke H J Higgs C et al. Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists[J]. Bioorganic & Medicinal Chemistry Letters 2010 20(8):2516-2519.
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